Intermediates :

 

Sr.No. API Intermediates
1 Adapalene 6-Bromo-2-Naphthoic acid methyl ester
2 Adapalene 2-(1-adamantyl)-4-Bromoanisole
3 Adapalene Anisole,2-4-(1-adamantyl)-4-bromo  
4 Adapalene 2-Naphthoic acid, 6 bromo, methyl ester 
5 Adapalene 1-Adamantanol 
6 Adapalene 4-Bromo-2-Adamantyl phenol
7 Amlexanox Ethoxymethylene Cyanoacetic acid ethyl ester
8 Amlexanox 4-Isopropyl phenol
9 Amorolfine Cis 2,6 Dimethyl morpholine
10 Anastrazole 1-Methyl-3, 5 Benzene Diacetonitrile
11 Anastrazole 5-(bromomethyl)-a,a,a,a-tetramethyl-1,3-benzenediacetonitrile 
12 Aripriprazole 7-(4-Bromobutoxy-3,4-Dihydro-2(IH) Qunilinone
13 Aripriprazole N-(2,3-Dichlorophenyl) Piperazine HCL
14 Atomoxetine N-MethylGamma-(2-Methylphenoxy) Benzenenpropanamine HCL
15 Atorvastatin (4R,Cis)-1,1-Dimethylethyl-cyanomethyl-2,2-Dimethyl-1,3-Dioxane-4-acetate
16 Atorvastatin (R)-4-Cyano-3-Hydroxybutyric acid ethyl ester
17 Azelastine 1-Methyl Azepin-4-One
18 Azelastine 2-[(4-chlorophenyl)acetyl]benzoice acid
19 Benazepril T-Butyl 3- S-amino-2,3,4,5-Tetrahydro-1H-[1]Benzepine-2-one-1-Acetate
20 Benazepril 1-Tetralone 
21 Benazepril 3-Bromo-2,3,4,5-Tetrahydro-1H-1-Benzazepine-2-one
22 Betamethasone series 16-β Methyl Epoxide
23 Bicalutamide 4-Cyano-3-Trifluoro Methyl Aniline 
24 Bicalutamide 4-Fluorothiophenol
25 Bisoprolol 4-Isopropoxyethoxymethyl-1-Hydroxybenzene 
26 Bosentan N-[6-chloro-5-(2-methoxyphenoxy)[2,2'-bipyrimidin]-4-yl]-4-(1,1-dimethylethyl)-Benzenesulfonamide
27 Candesartan Cyclohexyl-1-Chloro Ethyl Carbamate
28 Candesartan Methyl-2-(t-Butoxycarbonylamino)-3-Nitrobenzoate
29 Candesartan TritylChloride
30 Capecitabine 5'-Deoxy-2',3'-diacetoxy-5-fluorocytidine 
31 Carisoprodol 2-Methyl-2-Propyl-1,3-Propanediol
32 Carisoprodol 2-Methylvaleraldehyde
33 Cefditoren 4-Methyl-5-thiazolecarboxaldehyde
34 Cefpodoxime  Proxetil 1-Chloroethyl Isopropyl Carbonate
35 Cilastatin 7-Chloro-2-oxoheptanoic acid ethyl ester
36 Cilastatin (S)-2,2-Dimethylcyclopropanecarboxamide
37 Cilastatin L-Cysteine
38 Cinacalcet 3-Trifluoromethyl benzaldehyde
39 Cinacalcet (R)-(+)-1-(1-Naphthyl)-ethylamine
40 Dexamethsone series 16-α Methyl Epoxide
41 Docetaxel / Momentasone 4-Dimethylaminopyridine 
42 Dolasetron  Cis-1,4-Dichloro-2-Butene
43 Dolasetron / Indinavir N-Methylmorpholine-N-Oxide
44 Doxazosin 2-Chloro-4-Amino-6,7-Dimethoxy Quinazoline 
45 Duloxetine (S)-(-)-N-Dimethyl-3-Hydroxy-3-(2-Thienyl)-Propanamine
46 Duloxetine (S)-1-Hydroxy-1-(2-Thienyl)-3-Dimethylaminopropane
47 Duloxetine 2-Thienyl-2-Dimethylaminoethyl Ketone HCL
48 Epalrestat Rhodanine-3-Acetic acid
49 Epalrestat Trans-Alpha Cinnamaldehyde
50 Epinastine 6-aminomethyl-6,11-dihydro-5h-dibenz[b,e]azepine succinate
51 Ertapenem (4R,5S,6S)-3-(diphenyloxy)phosphoryloxy-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3,2,0]hept-2-ene-2-carboxylate.
52 Ertapenem (2S,4S) -2-[(3-carboxyphenyl)aminocarbonyl]-4-thio-1- (p-nitrobenzyloxycarbonyl)-1-pyrrolidine
53 Ertapenem [3S(S),4R]-4-acetoxy-3-[1-(tert-butyldimethylsiloxy)ethyl]-2-azetidino
54 Etodolac 3-Ketovaleric acid methyl ester
55 Etodolac 7-Ethyl Trytophol
56 Etodolac 7-Ethyl-3-[2-Hydroxyethyl) Indole
57 Etodolac Etodolac methyl ester
58 Faropenem Ally(1'R,2'''R,5R,6S)-6(1'-tert-butyl dimethyl silyloxyethy)-2-(2''-tetrahydrofuranyl)penem-3-carboxylate
59 Faropenem Sodium-2-ethyl Hexanoate
60 Faropenem Tetrabutyl Ammonium Fluoride
61 Fexofenadine a,a-Diphenyl-4-piperidinemethanol
62 Fexofenadine Ethyl,4-(4-chloro-1-oxobutyl)-a,a-dimethylbenzene acetate
63 Fexofenadine Ethyl,4-(4-[hydroxydiphenylmethyl-1-piperidinyl]-1-oxbutyl)-a,a dimethylbenzene acetate hcl
64 Formoterol  R-4-Benzyloxy-3-Nitro Phenyl Oixrane  
65 Gemcitabine Acetyl Cytosine
66 Gemcitabine Dimethylamino Pyridine
     
67 Gemcitabine Ethyl Bromo Difluoro acetate
68 Gemcitabine 3,5-Bis(benzoyl)-2-Desoxy-2,2-Difluoro-1-oxoribose 
69 Gemcitabine 3,5-Bis(benzoyl)-1-methanesulfonyl;oxy-2-desoxy-2,2-difluororibose 
70 Gemcitabine 2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dibenzoate (GN-9)
71 Gemfibrozil Isobutyl 5-chloro-2,2-dimethylvalerate 96%min
72 Gemfibrozil Methyl 5-chloro-2,2-dimethyl valerate 95%min
73 Gliclazide 3-Amino-3-Azabicyclo[3,3,0]Octane
74 Glimepiride 4-(2-(3-Ethyl-4-2-oxo-3-Pyrolline-1-Ccarboxamido)Ethyl Benzene Sulfonamide 
75 Glimepride Trans-4-Methyl Cyclo Hexane Isocyanate
76 Granisteron 1-Methylindazole-3-Carboxylic Acid - 10 kgs
77 Granisteron Endo-9-Methyl-9-Azabicyclo[3,3,1] nonane-3-Amine
78 Ibandronate Sodium 3-(N-methyl-N-pentylamino)-propionic acid Hcl
79 Imatinib Mesylate Cynamide solution
80 Imiquimod 1H-Imedazo[4,5-c]quinoline,4-chloro-1-(2-methylpropyl) 
81 Imiquimod Quinoline,3-amino-4-(2-methylpropylamino)                  
82 Imiquimod/ Dolasetron  Trifluoroacetic Anhydride
83 Irbesartan Bromo OTBN 
84 Irinotecan 4-Piperidinopiperidine
85 Lercanidipine 1-(3,3-Diphenyl-N-Methylpropylamino)-2-Methyl-2-Propanol 
86 Lercanidipine 2,6-dimethyl-5-methoxy carbonyl-4-(3-nitro phenyl_-1,4 dihydropyridine -3-carboxylic Acid
87 Lercanidipine 2,6-dimethyl-5-methoxy carbonyl-4-(3-nitro phenyl-1,4 dihydro pyridine)-3-carboxylic Acid
88 Lercanidipine 1-(3,3-Diphenyl-N-Methylpropylamino)-2-Methyl-2-Propanol
89 Letrozole 4-Fluorobenzonitrile
90 Letrozole Alpha-Bromo Tolunitrile
91 Letrozole Potassium-Tert-Butoxide
92 Letrozole 4,4-(Hydroxymethylene)bisbenzonitrile 
93 Levitiracetam Alpha-[2-(Methylthio)Ethyl]-2-Oxo-1-Pyrrolidineacetamide
94 Levosulpiride 2-S-(Aminomethyl)-1-Ethyl Pyrrolidine
95 Levosulpiride 5-(chlorosulfonyl)-2-methoxy benzoic acid
96 Levothyroxine N-Acetyl-3,5-Diiodo-L-Tyrosine
97 Lisinopril Lisinopril ester (CAS No. 103300-91-0) 30% solution
98 Lisinopril L-Proline benzyl Ester HCL
99 Lisinopril N2-[(1S)-ethoxycarbonyl-3-pheynlpropyl]-N6-trifluoroacetyl-L-lysine
100 Lisinopril N-6-Trifluoro Acetyl – L – Lysine
101 Mebhydroline 1-Benzyl-1-phenylhydrazine hydrochloride
102 Mefloquin 2-Trifluoromethylaniline
103 Meloxicam 2-Amino-5-Methylthiazole 
104 Memantine 1,3-Dimethyl Adamantine
105 Mifepristone Estra-4,9-diene-3,17-dion
106 Mirtazapine 1-methyl-3-phenyl piperazine (98.0%min)
107 Mirtazapine 2-Chloro-3-Cyano Pyridine
108 Mitoxantrone 1,4,5,8-tetrahydroxyanthraquinone
109 Nateglinide D-Phenyl Alanaine Methyl Ester HCL
110 Ofloxacin Ofloxacin Quinolinic Acid
111 Olmesartan 4-(1-Hydroxyisopropyl)-2-propyl-1-{{2'-[1-(triphenylmethyl)-5-tetrazolyl][1,1'-biphenyl]-4-yl}-methyl}-5-imidazolecarboxylic acid (5-methyl-2-oxo-1,3-dioxol-4-yl)-methyl ester
112 Oseltamivir Shikimic acid
113 Oseltamivir (1S,5R,6S)-5-(1-ethylpropoxy)-7-oxobicyclo[4,1,0]hept-3-ene-3-carboxylic acid ethyl ester
114 Palonosetron 3-Quinuclidinone HCL
115 Paroxetine 3-S Trans (-3-[1,3 Benzodioxol-5-Yloxy) Methyl-]4'(4-Fluoro Phenyl)N-Methyl Piperidine 
116 Paroxetine Trans (+)-1-Methyl-Y-(Para Fluoro phenyl)Piperidine-3-carbinol 99%min 
117 Perindopril (2S,3aS,7aS)-2-Carboxyoctahydroindole 
118 Perindopril (S)-indoline-2-carboxylic acid
119 Perindopril L-Norvaline 
120 Perindopril L-octahydroindole-2-carboxylic acid
121 Perindopril N-[1-(S)-(Ethoxycarbonyl)Butyl]-(S)-Alanine
122 Pramipexole (6S)-4,5,6,7-Tetrahydro-1,3-benzothiazole-2,6-diamine
123 Pramipexole (S)-2-Amino-6-propylamino-4,5,6,7-tetrahydrobenzthiazole
124 Pramipexole 4-(Phthalimido)-Cyclohexanone  
125 Prostaglandin F2 Alfa Hexamethyl Phosphoramide
126 Quetiapine  Dibenzo [b,f][1,4]Thiazepine-11-[10H]one
127 Quetiapine  Piperazine,4-[2-(2-hydroxyethoxy) ethyl 
128 Quetiapine Fumarate 2-(2-Chloroethoxy) Ethanol
129 Quinapril Ethyl-2-oxo-4-Phenyl Butyrate
130 Quinapril / Enalapril N-(1-S-Carbethoxy-3-Phenylpropyl)-S-Alanine
131 Raloxifene 4[2-(1-Piperidinyl)Ethoxy]Benzoic Acid HCL
132 Raloxifene 6-methoxy-2-(4-methoxy phenyl)benzo(b) thiophene
133 Repaglinide 2-Fluorobenzaldehyde
134 Repaglinide 4-(ethoxycarbonyl)3-ethoxyphenylacetic acid
135 Repaglinide (S)-[A-(2-methylpropyl)-2-(1-piperidinyl)benzene-methanamine 
136 Resiperidone 3-(2-Chloroethyl)-6,7,8,9-Tetrahydro-2-Methyl-4H-Pyrido [1,2-a] Pyrimidine-4-One
137 Resiperidone 4-(2,4-Difluorophenyl)-4-Piperidinyl-Methanone Hcl
138 Rimonabant 5-(4-chlorophenyl-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxylic acid
139 Risperidone  6-fluoro-3-(piperidin-4-yl)benzo[d]isoxazole
140 Rivastigmine DI Para Toluyl D-Tartaric acid 
141 Ropinirole 4-(2-Hydroxyethyl) oxyindole
142 Ropinirole 4-[2-(benzoate)ethyl]-3-Chloro Oxyindole
143 Ropinirole (2-Methyl-3-Nitrophenyl) N,N-Dipropylacetamide
144 Ropinirole 2-Methyl-3-nitro phenyl acetic acid
145 Rosuvastatin 4-(4-fluorophenyl)-6-isopropyl-2-(N-Methyl-N-methylsulphonylamino)-5-pyrimidinecarboxaldehyde
146 Sultamicillin Chloroiodomethane
147 Tamsulosin 2-(O-EthoxyPhenoxy)Ethyl Bromide
148 Tamsulosin 5-Acetonyl-2-Methoxybenzene Sulfonamide
149 Tamsulosin R-(-)-5-[2(2-Amino-2-Methyl)Ethyl]-2-Methoxybenzene Sulfonamide
150 Tazarotene 6-Chloronicotinic acid
151 Tazarotene Diethyl Chlorophosphate
152 Tazarotene Lithium Diisopropylamine
153 Tazarotene Prenyl Bromide
154 Telithromycin N-(3-Dimethylamino)propyl-N'-ethylcabidiimide
155 Telithromycin N-(3-Dimethylamino)propyl-N'-ethylcabidiimide
156 Telithromycin Methane Sulfonic Anhydride
157 Terazosin 2-Chloro-4-Amino-6,7-Dimethoxy Quninazoline
158 Terazosin N-(Tetrahydro-2-Furoyl)-piperazine HBr
159 Ticarcillin Diisopropyl Ether
160 Ticarcillin 3-Thiophene Malonic acid
161 Tirofiban N-(Butyl Sulfonyl)-L-Tyrosine  97%min
162 Tirofiban 4-(4-Chlorobutyl) pyridine  97%min
163 Torasemide 4-(3-Methylphenyl)-Amino-3-Pyridine Sulfonamide 
164 Trimebutine 2-Dimethylamino-2-Phenyl-1-Butanol
165 Trioxsalen 2-Methylresorcinol 
166 Tropisetron/ Dolasetron 3-Indolecarboxylic acid 
167 Valsartan L-Valine Methyl ester Hydrochloride
168 Voriconazole  (2R,3S/2S,3R)-2-(2,4-difluorophenyl)-3-(5-fluoro-4-pyrimidinyl)-1-(1H-1,2,4-triazol-1-yl) -2-butanol (n-1)
169 Voriconazole  (2R,3S/2S,3R)-3-(4-Chloro-5-Fluoro-6-Pyrimidinyl)-2-(2,4-Difluorophenyl)-1-(1H-1,2,4-Triazol-1-yl)-2-Butanol HCL (N-2)
170 Zanamavir N-Acetylneuraminic acid
171 Zoledronic acid 1H-imidazole-1-acetic acid 
172 Zonisamide 1,2-Benzisoxazole-3-Methane Sulfonate Sodium
 
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